Catalog / N-[3-氟-1-(羟甲基)环丁基]氨基甲酸叔丁酯

N-[3-氟-1-(羟甲基)环丁基]氨基甲酸叔丁酯

tert-Butyl N-[3-fluoro-1-(hydroxymethyl)cyclobutyl]carbamate
Molecular Structure
CAS Number
1232365-48-8
Molecular Formula
C10H18FNO3
Molecular Weight
219.25
Purity
≥95%
InChIKey
MLIXJRTXFCDVNT-UHFFFAOYSA-N
SMILES
CC(C)(C)OC(=O)NC1(CC(C1)F)CO
Appearance
Solid (predicted)
Storage
Store at 2-8°C
Description

tert-Butyl N-[3-fluoro-1-(hydroxymethyl)cyclobutyl]carbamate is a Boc-protected fluorocyclobutane building block with a hydroxymethyl group. Used as a pharmaceutical intermediate for introducing fluorinated cyclobutane motifs into drug candidates, offering enhanced metabolic stability and modified lipophilicity.

Applications

Pharmaceutical intermediate; medicinal chemistry; cyclobutane building block

Ordering

Packaging: 100 mg; 250 mg; 1 g; 5 g

Availability

Status Check Availability
Purity ≥95%
Grade Research grade
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